Dorzolamide

Mechanism of action:
Dorzolamide is a carbonic anhydrase inhibitor. Carbonic anhydrase II is present in the epithelial cells of the ciliary body of the eye and catalyzes the formation of bicarbonate (HCO₃⁻), which is an essential component in aqueous humor production. By inhibiting carbonic anhydrase II, dorzolamide reduces aqueous humor secretion and lowers intraocular pressure.
Reference(s):
1. Martens-Lobenhoffer J et al. (2002). Clinical pharmacokinetics of dorzolamide. Clin Pharmacokinet.
2. Balfour JA et al. (1997). Dorzolamide. A review of its pharmacology and therapeutic potential in the management of glaucoma and ocular hypertension. Drugs Aging.
3. Arieta C et al. (2002). Dorzolamide versus apraclonidine in the prevention of the intraocular pressure spike after Nd:YAG laser posterior capsulotomy. Curr Eye Res.
