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Eslicarbazepine

艾司利卡西平

Mechanism of action:

Eslicarbazepine 會選擇性地與處於失活狀態的鈉離子通道(sodium channel)結合,延長通道恢復至可開啟狀態的時間,使神經元在高頻刺激下無法持續產生動作電位,降低神經元過度放電的機率。

​Reference(s):

Tian M et al. (2014). Carbamazepine derivatives with P2X4 receptor-blocking activity. Bioorg Med Chem.

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