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Fluocinonide

醋酸氟輕松
Mechanism of action:
Fluocinonide 是一種高效力外用糖皮質類固醇(high-potency topical corticosteroid),屬於合成氟化類固醇(fluorinated corticosteroid)衍生物。Fluocinonide 穿透皮膚進入細胞後,與細胞質中的糖皮質類固醇受體(glucocorticoid receptor)結合,形成藥物-受體複合體並進入細胞核,提升抗發炎基因(如 annexin A1)表達;抑制發炎轉錄因子(如 NF-κB、AP-1)等。
Reference(s):
1. Jessop S et al. (2001). Drugs for discoid lupus erythematosus. Cochrane Database Syst Rev.
2. Zhou Y et al. (2024). TTD: Therapeutic Target Database describing target druggability information. Nucleic Acids Res.
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