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Mafenide

磺胺米隆
Mechanism of action:
Mafenide 是一種磺胺類(sulfonamide)分子。Mafenide 會和對胺基苯甲酸(4-Aminobenzoic acid,PABA)競爭,抑制細菌二氫蝶酸合酶(dihydropteroate synthase),使二氫葉酸(dihydrofolic acid)生成下降,進而阻斷四氫葉酸(tetrahydrofolic acid)的生成,導致細菌的 DNA、RNA 與蛋白質生成受阻。
Reference(s):
Maghsoudi H et al. (2011). Comparison between topical honey and mafenide acetate in treatment of burn wounds. Ann Burns Fire Disasters.
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