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Moricizine

莫雷西嗪
Mechanism of action:
Moricizine 能抑制心肌細胞膜上的快速鈉離子通道(fast sodium channel),減緩去極化(depolarization),降低心肌的傳導速度。
Reference(s):
1. Ahmmed GU et al. (2002). Analysis of moricizine block of sodium current in isolated guinea-pig atrial myocytes. Atrioventricular difference of moricizine block. Vascul Pharmacol.
2. Chen X et al. (2002). TTD: Therapeutic Target Database. Nucleic Acids Res.
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