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Tacrine

他克林

Mechanism of action:

Tacrine 是一種乙醯膽鹼酯酶抑制劑(acetylcholinesterase inhibitor),屬於四氫氨基吖啶(tetrahydroaminoacridine)衍生物。Tacrine 能可逆性抑制乙醯膽鹼酯酶(acetylcholinesterase),減少突觸間隙中乙醯膽鹼(acetylcholine)的分解速度,增強膽鹼性神經傳導。

​Reference(s):

Qizilbash N et al. (1998). Cholinesterase inhibition for Alzheimer disease: a meta-analysis of the tacrine trials. Dementia Trialists' Collaboration. JAMA.

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